生物活性
Bisoprolol fumarate是一种属于β受体阻滞剂的药物，β受体阻滞剂是一类主要用于心血管疾病的药物。更具体地说，它是一种选择性的β1肾上腺素能受体阻滞剂。
靶点信息
化学数据
| 目录号 | A10149 |
| 作用机制 | Blocker (阻断剂) |
| M. Wt | 441.5 |
| Formula | C22H35NO8 |
| Purity | >99% |
| Storage | Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles. |
| CAS No. | 104344-23-2 |
| Synonyms | Zebeta |
| SMILES | CC(C)NCC(COC1=CC=C(C=C1)COCCOC(C)C)O.C(=C/C(=O)O)\C(=O)O |
溶解度
| In vitro | DMSO | 76 mg/mL (172.13 mM) |
| Water | 76 mg/mL (172.13 mM) |
| Ethanol | 76 mg/mL (172.13 mM) |
*<1 mg/ml means slightly soluble or insoluble.
*Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
储备液配制
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
| 0.1 mM | 22.65 mL | 113.25 mL | 226.5 mL |
| 0.5 mM | 4.53 mL | 22.65 mL | 45.3 mL |
| 1 mM | 2.27 mL | 11.33 mL | 22.65 mL |
| 5 mM | 0.45 mL | 2.27 mL | 4.53 mL |
*The above data is based on the productmolecular weight 441.5 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
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