LAS191954 是有效的、选择性的、口服有效的 PI3Kδ 的抑制剂，可用于炎症相关疾病的研究，其 IC50 值为 2.6 nM。
CAS：1403947-26-1
分子式：C20H15N9O
分子量：397.39
纯度：98%
存储：Store at -20°C

Background:

LAS191954 is a potent, selective and orally active PI3Kδ inhibitor for inflammatory diseases treatment, with an IC50 of 2.6 nM[1]. PI3Kδ|2.6 nM (IC50)

[1]. Erra M, et al. Discovery of a Potent, Selective, and Orally Available PI3Kδ Inhibitor for the Treatment of Inflammatory Diseases. ACS Med Chem Lett. 2016 Nov 30;8(1):118-123.