生物活性
Bupivacaine HCl与化学相关的局部麻醉药相比,Bupivacaine HCl是一种更有效的cAMP抑制剂,较不易产生心血管毒性。
靶点信息
化学数据
目录号 | A10168 |
M. Wt | 324.9 |
Formula | C18H28N2O.HCl |
Purity | >99% |
Storage | Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for36 months. In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles. |
CAS No. | 18010-40-7 |
Synonyms | Marcain, Marcaine, Sensorcaine, Vivacaine |
SMILES | CCCCN1CCCCC1C(=O)NC2=C(C=CC=C2C)C.Cl |
溶解度
In vitro | DMSO | 60 mg/mL (184.67 mM) |
Water | 21 mg/mL (64.63 mM) |
Ethanol | 60 mg/mL (184.67 mM) |
*<1 mg/ml means slightly soluble or insoluble. *Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
储备液配制
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
0.1 mM | 30.78 mL | 153.89 mL | 307.79 mL |
0.5 mM | 6.16 mL | 30.78 mL | 61.56 mL |
1 mM | 3.08 mL | 15.39 mL | 30.78 mL |
5 mM | 0.62 mL | 3.08 mL | 6.16 mL |
*The above data is based on the productmolecular weight 324.9 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.