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Naftopidil(Flivas)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Naftopidil(Flivas)图片
CAS NO:57149-07-2
包装与价格:
包装价格(元)
250mg电议
10mM * 1mL in DMSO电议

产品名称
KT-611, BM-15275
产品介绍

生物活性

Naftopidil (Flivas)是选择性的α1-肾上腺素能受体拮抗剂或α受体阻滞剂,Ki为58.3 nM。

靶点信息

α1D-adrenergic receptorα1A-adrenergic receptorα1B-adrenergic receptor
1.2 nM(Ki)3.7 nM(Ki)20 nM(Ki)

化学数据

目录号A10618
M. Wt465.41
FormulaC24H28N2O3.2HCl
Purity>99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No.57149-07-2
SynonymsKT-611, BM-15275
SMILESCOC1=CC=CC=C1N2CCN(CC2)CC(COC3=CC=CC4=CC=CC=C43)O

溶解度

In vitroDMSO77 mg/mL (196.17 mM)
WaterInsoluble
EthanolInsoluble
*<1 mg/ml means slightly soluble or insoluble.
*Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

储备液配制

Concentration / Solvent Volume / Mass1 mg5 mg10 mg
0.1 mM21.49 mL107.43 mL214.86 mL
0.5 mM4.3 mL21.49 mL42.97 mL
1 mM2.15 mL10.74 mL21.49 mL
5 mM0.43 mL2.15 mL4.3 mL

*The above data is based on the productmolecular weight 465.41. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.