TTA-Q6是一种选择性的T型钙离子通道(Ca2+channel)拮抗剂,可用于神经领域的研究。
CAS:910484-28-5
分子式:C20H15ClF3N3O
分子量:405.8
纯度:98%
存储:Store at -20°C
Background:
TTA-Q6 is a selective T-type Ca2+ channel antagonist, used in the neurological disease.
TTA-Q6 is a selective T-type Ca2+ channel antagonist, with 14 nM and 590 nM in FLIPR depolarized assaay and FLIPR hyperpolarized assay[1].
[1]. Schlegel KA, et al. Discovery and expanded SAR of 4,4-disubstituted quinazolin-2-ones as potent T-type calcium channel antagonists. Bioorg Med Chem Lett. 2010 Sep 1;20(17):5147-52.