Molibresibbesylate(GSK525762C;I-BET762besylate)是BET溴结构域抑制剂,IC50为32.5-42.5nM。
CAS:1895049-20-3
分子式:C28H28ClN5O5S
分子量:582.07
纯度:98%
存储:Store at -20°C
Background:
Molibresib besylate (GSK 525762C; I-BET 762 besylate) is a BET bromodomain inhibitor with IC50 of 32.5-42.5 nM.
IC50: 32.5-42.5 nM (BET)[1]
[1]. Nicodeme E, et al. Suppression of inflammation by a synthetic histone mimic. Nature. 2010 Dec 23;468(7327):1119-23.