c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm 是一种有效选择性的、短效肽的 V2 受体 (V2R) 激动剂,对 hV2R 和rV2R EC50 值分别为 0.25 和 0.05 nM。
CAS:1647119-71-8
分子式:C47H69ClN12O9S2
分子量:1045.71
纯度:98%
存储:Store at -20°C
Background:
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm is a is a potent, selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.25 and 0.05 nM for hV2R and rV2R, respectively[1].
EC50: 0.25 nM (hV2R), 0.05 nM (rV2R)[1]
[1]. Wi?niewski K, et al. Discovery of Potent, Selective, and Short-Acting Peptidic V2 Receptor Agonists. J Med Chem. 2019 May 23;62(10):4991-5005.