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Acevaltrate
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Acevaltrate图片
CAS NO:25161-41-5
规格:98%
分子量:480.5
包装与价格:
包装价格(元)
5mg电议
10mg电议
25mg电议
50mg电议
100mg电议

产品介绍
Acevaltrate从Valerianaglechomifolia中分离,抑制大鼠肾和脑半球中Na+/K+-ATP酶活性,IC50分别为22.8±1.1μM和42.3±1.0μM。
CAS:25161-41-5
分子式:C24H32O10
分子量:480.5
纯度:98%
存储:Store at -20°C

Background:

Acevaltrate, isolated from Valeriana glechomifolia, inhibits the Na+/K+-ATPase activity in the rat kidney and brain hemispheres with IC50s of 22.8±1.1 μM and 42.3±1.0 μM, respectively[1].


Acevaltrate differentiallys inhibit the activity of rat P-type ATPases in vitro. 60.7±7.3% inhibition of the rat H+/K+-ATPase is achieved at 100 µM[1].



[1]. Bettero GM, et al. In vitro effect of valepotriates isolated from Valeriana glechomifolia on rat P-type ATPases. Planta Med. 2011 Oct;77(15):1702-6.