OT-Rantagonist2是一种非肽类OT-R拮抗剂,抑制大鼠催产素受体（IC50=0.33μM）。
CAS：364071-16-9
分子式：C28H29N3O4
分子量：471.55
纯度：98%
存储：Store at -20°C

Background:

OT-R antagonist 2 is a nonpeptide low molecular weight OT-R antagonist. OT-R antagonist 2 inhibitis IP3-Synthesis, rat OT-R (IC50 = 0.33 μM).IC50 value: 0.33μMTarget: oxytocin receptor

[1]. Cirillo R, et al. Pharmacology of (2S,4Z)-N-[(2S)-2-hydroxy-2-phenylethyl]-4-(methoxyimino) -1-[(2’-methyl[1,1’-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide, a new potent and selective nonpeptide antagonist of the oxytocin receptor. J Pharmacol Exp T [2]. William Nadler, et al. Method for preparing pyrrolidine oximes. WO/2005082848/A2. [3]. Serge Halazy, et al. Pharmaceutically active pyrrolidine derivatives as bax inhibitors.WO/2001074769/A1. [4]. Serge Halazy, et al. Pharmaceutically active pyrrolidine derivatives as bax inhibitors. WO/2001072705/A1.