CBP/P300bromodomaininhibitor-3是CBP/P300溴结构域家族的有效抑制剂。CBP/P300bromodomaininhibitor-3抑制CBP(IC50=0.01-0.1µμ)和BRD4(IC50=1-1000µμ)活性。
货号:ajcx30344
CAS:2304416-91-7
分子式:C27H31N3O4
分子量：461.55
溶解度:DMSO: 200 mg/mL (433.32 mM)
纯度：98%
存储：Store at -20°C
库存：现货

Background:

CBP/P300 bromodomain inhibitor-3 is a potent inhibitor of the CBP/P300 family of bromodomains. CBP/P300 bromodomain inhibitor-3 inhibits CBP (IC50=0.01-0.1 µμ) and BRD4 (IC50=1-1000 µμ) activity[1].

[1]. Shawn E.R. Schiller, et al. Tetrahydro-imidazo quinoline compositions as cbp/p300 inhibitors. WO2019055877A1.