Axitinib-d3 是氘标记的 Axitinib。Axitinib 是多靶点的酪氨酸激酶抑制剂，抑制 VEGFR1，VEGFR2，VEGFR3， PDGFRβ 的 IC50 值分别为4，20，4，2 nM。
货号:ajcx33222
CAS:1126623-89-9
分子式:C22H15D3N4OS
分子量：389.49
溶解度:N/A
纯度：98%
存储：Store at -20°C
库存：现货

Background:

Axitinib-d3 (AG-013736-d3) is deuterium labeled Axitinib. Axitinib is a multi-targeted tyrosine kinase inhibitor with IC50s of 0.1, 0.2, 0.1-0.3, 1.6 nM for VEGFR1, VEGFR2, VEGFR3 and PDGFRβ, respectively.

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