(3R,4R)-A2-32-01 (compound 2),抗毒力药物,是一种特异性的酪蛋白溶解蛋白蛋白酶 (ClpP) 抑制剂,EC50 值为 4.5 μM,并显示出可耐受的细胞毒性。
货号:ajcx16134
CAS:1359752-95-6
分子式:C19H27NO2
分子量:301.42
溶解度:DMSO: 200 mg/mL (663.53 mM)
纯度:98%
存储:Store at -20°C
库存:
现货Background:
(3R,4R)-A2-32-01 (compound 2), an anti-virulence drug, is a specific caseinolytic protein proteases (ClpP) inhibitor with an EC50 of 4.5 μM, and shows a tolerable cytotoxicity[1].
[1]. Zeiler E, et al. Development and characterization of improved β-lactone-based anti-virulence drugs targetingClpP. Bioorg Med Chem. 2012 Jan 15;20(2):583-91.