TFA salt of virodhamine, an endogenous cannabinoid receptor mixed agonist/antagonist
货号:ajcx27028
CAS:1415264-56-0
分子式:C22H37NO2.CF3CO2H
分子量:461.56
溶解度:Soluble in DMSO
纯度:98%
存储:Store at -20°C
库存:
现货Background:
TFA salt of virodhamine, an endogenous cannabinoid receptor mixed agonist/antagonist that is found in higher concentrations peripherally than anandamide. Virodhamine is a full agonist at GPR55 and CB2 and partial agonist/antagonist at CB1 (EC50 values are 12, 381 and 2920 nM at GPR55, CB2 and CB1 receptors respectively).
Porter et al (2002) Characterization of a novel endocannabinoid, virodhamine, with antagonist activity at the CB1 receptor. J.Pharmacol.Exp.Ther. 301 1020 PMID:12023533