Propofol 有效直接地激活 GABAA 受体和抑制谷氨酸受体介导的兴奋性突触传递。Propofol 具有抗伤害感受特性，可用于镇静和催眠。
货号:ajcx16606
CAS:2078-54-8
分子式:C12H18O
分子量：178.27
溶解度:DMSO: 100 mg/mL (560.95 mM); H2O: 1 mg/mL (5.61 mM)
纯度：98%
存储：Store at -20°C
库存：现货

Background:

Propofol potently and directly activates GABAA receptor and inhibits glutamate receptor mediated excitatory synaptic transmission. Propofol has antinociceptive properties and is used for sedation and hypnotic[1].

[1]. R Nadeson, et al. Antinociceptive Properties of Propofol: Involvement of Spinal Cord Gamma-Aminobutyric acid(A) Receptors. J Pharmacol Exp Ther . 1997 Sep;282(3):1181-6.