GCPII-IN-1 TFA 是一种谷氨酸羧肽酶 II (GCPII; PSMA) 抑制剂支架,Ki 为 44.3 nM。
货号:ajcx35486
CAS:1269794-89-9
分子式:C14H22F3N3O9
分子量:433.33
溶解度:H2O : 160 mg/mL (369.23 mM; Need ultrasonic)
纯度:98%
存储:Store at -20°C
库存:
现货Background:
GCPII-IN-1 TFA is a glutamate carboxypeptidase II (GCPII, or PSMA) inhibitor scaffold with a Ki of 44.3 nM[1].
[1]. Jan Tykvart, et al. Rational design of urea-based glutamate carboxypeptidase II (GCPII) inhibitors as versatile tools for specific drug targeting and delivery. Bioorg Med Chem. 2014 Aug 1;22(15):4099-108.