GSK251 是一种高效、高选择性、口服生物利用度的 PI3Kδ 抑制剂，具有新颖的结合模式。
货号:ajcx37952
CAS:2125968-05-8
分子式:C29H37FN6O4S
分子量：584.71
溶解度:DMSO : 62.5 mg/mL (106.89 mM; ultrasonic and warming and heat to 60°C)
纯度：98%
存储：Store at -20°C
库存：现货

Background:

GSK251 is a highly potent, highly selective, orally bioavailable inhibitor of PI3Kδ with a novel binding mode.

[1]. Down K, et al. Discovery of GSK251: A Highly Potent, Highly Selective, Orally Bioavailable Inhibitor of PI3Kδ with a Novel Binding Mode. J Med Chem. 2021 Sep 23;64(18):13780-13792.