Cerlapirdine (SAM-531, PF-05212365) 是一种选择性和有效的 5-羟色胺 6 (5-HT6) 受体的完全拮抗剂。Cerlapirdine 具有研究阿尔茨海默病的潜力。
货号:ajcx36700
CAS:925448-93-7
分子式:C22H23N3O3S
分子量：409.5
溶解度:DMSO : 41.67 mg/mL (101.76 mM; ultrasonic and warming and adjust pH to 3 with HCl and heat to 60°C)
纯度：98%
存储：Store at -20°C
库存：现货

Background:

Cerlapirdine (SAM-531, PF-05212365) is a selective and potent full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine has the potential for researching the Alzheimer’s disease[1].

[1]. Tse S, et al. Disposition and metabolic profiling of [(14)C]cerlapirdine using accelerator mass spectrometry. Drug Metab Dispos. 2014;42(12):2023-2032.