Stafib-1 is the first small molecule inhibitor of the STAT5b SH2 domain (Ki =44 nM) with more than 50-fold selectivity over STAT5a. References: Elumalai N, Natarajan K, Berg T. Halogen-substituted catechol bisphosphates are potent and selective inhibitors of the transcription factor STAT5b. Bioorg Med Chem. 2017 Jul 15;25(14):3871-3882. doi: 10.1016/j.bmc.2017.05.039. Epub 2017 May 18. PubMed PMID: 28559059.
纯度:≥98%
CAS:1688703-26-5