L-152,804 is a potent, selective non-peptide neuropeptide Y Y5 receptor antagonist (Ki = 26 nM for hY5). L-152,804 exhibits > 300-fold selectivity over hY1, hY2, and hY4 receptors. References: Long M, Zhou J, Li D, Zheng L, Xu Z, Zhou S. Long-Term Over-Expression of Neuropeptide Y in Hypothalamic Paraventricular Nucleus Contributes to Adipose Tissue Insulin Resistance Partly via the Y5 Receptor. PLoS One. 2015 May 18;10(5):e0126714. doi: 10.1371/journal.pone.0126714. PubMed PMID: 25993471; PubMed Central PMCID: PMC4436377.
纯度:≥98%
CAS:6508-43-6