GZ-793A inhibits dopamine uptake at the vesicular monoamine transporter-2 (VMAT2. A lobelane analogue, GZ-793A interacts with the vesicular monoamine transporter-2 to inhibit the effect of methamphetamine. References: Penthala NR, Ponugoti PR, Nickell JR, Deaciuc AG, Dwoskin LP, Crooks PA. Pyrrolidine analogs of GZ-793A: synthesis and evaluation as inhibitors of the vesicular monoamine transporter-2 (VMAT2). Bioorg Med Chem Lett. 2013 Jun 1;23(11):3342-5. doi: 10.1016/j.bmcl.2013.03.092. Epub 2013 Apr 2. PubMed PMID: 23597792; PubMed Central PMCID: PMC3725993.
纯度:≥98%
CAS:1356447-90-9