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TRV130 HCl(Oliceridine)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
TRV130 HCl(Oliceridine)图片
CAS NO:1401031-39-7
包装与价格:
包装价格(元)
5mg电议
10mg电议
25mg电议

产品名称
TRV-130, TRV 130
产品介绍

生物活性

TRV130 HCl (Oliceridine)是一种新型的μ-opioid 受体(MOR)G蛋白偏向配体。诱导强大的G蛋白信号传导(pEC50 = 8.1),效力和功效与吗啡相似,但β-arrestin募集和受体内在化作用要低得多。

化学数据

目录号A15444
作用机制Agonist (激动剂)
M. Wt423.01
FormulaC22H31ClN2O2S
Purity>99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No.1401031-39-7
SynonymsTRV-130, TRV 130
SMILESCOC1=C(SC=C1)CNCCC2(CCOC3(C2)CCCC3)C4=CC=CC=N4.Cl

储备液配制

Concentration / Solvent Volume / Mass1 mg5 mg10 mg
0.1 mM23.64 mL118.2 mL236.4 mL
0.5 mM4.73 mL23.64 mL47.28 mL
1 mM2.36 mL11.82 mL23.64 mL
5 mM0.47 mL2.36 mL4.73 mL

*The above data is based on the productmolecular weight 423.01. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.