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SR9243
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
SR9243图片
CAS NO:1613028-81-1
包装与价格:
包装价格(元)
10mg电议
25mg电议
50mg电议

产品名称
SR-9243, SR 9243
产品介绍

生物活性

SR9243是有效的选择性LXR反向激动剂。SR9243通过抑制脂质产生和Warburg效应杀死癌细胞。它在多种类型的癌症中诱导细胞死亡,并且不会引起副作用,而这些副作用已使先前针对这些过程的尝试脱轨。

靶点信息

LXR

化学数据

目录号A15535
作用机制Agonist (激动剂)
M. Wt626.62
FormulaC31H32BrNO4S2
Purity>99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No.1613028-81-1
SynonymsSR-9243, SR 9243
SMILESCC(C=C(C)C=C1C)=C1S(N(CC2=CC=C(C3=CC(C)=CC=C3)C=C2)CCC4=CC=CC(Br)=C4)(=O)=O.O=S=O

溶解度

In vitroDMSOInsoluble
WaterInsoluble
EthanolDMF: Warmed: 87 mg/mL (138.84 mM)
*<1 mg/ml means slightly soluble or insoluble.
*Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

储备液配制

Concentration / Solvent Volume / Mass1 mg5 mg10 mg
0.1 mM15.96 mL79.79 mL159.59 mL
0.5 mM3.19 mL15.96 mL31.92 mL
1 mM1.6 mL7.98 mL15.96 mL
5 mM0.32 mL1.6 mL3.19 mL

*The above data is based on the productmolecular weight 626.62. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.