| CAS NO: | 1671088-84-8 |
| 包装 | 价格(元) |
| 100 μg | 电议 |
| 250 μg | 电议 |
| 500 μg | 电议 |
| 1mg | 电议 |
| Cas No. | 1671088-84-8 |
| Canonical SMILES | ClC1=CC=CC=C1C2=CC=CC(CN3C(NC(CCCNC(CCl)=N)C3=O)=O)=C2 |
| 分子式 | C21H22Cl2N4O2 |
| 分子量 | 433.3 |
| 溶解度 | DMF: 30 mg/ml,DMSO: 30 mg/ml,DMSO:PBS (pH 7.2) (1:1): 0.5 mg/ml,Ethanol: 10 mg/ml |
| 储存条件 | Store at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
| 产品描述 | CAY10727 is an inhibitor of protein arginine deiminase 3 (PAD3; kinact/KI= 15,600 M-1min-1).1It is selective for PAD3 over PAD1, -2, and -4 (kinact/KIs = 360, 1,110, and 1,460 M-1min-1, respectively). 1.Jamali, H., Khan, H.A., Stringer, J.R., et al.Identification of multiple structurally distinct, nonpeptidic small molecule inhibitors of protein arginine deiminase 3 using a substrate-based fragment methodJ. Am. Chem. Soc.137(10)3616-3621(2015) |
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