TP-064 是一种有效的选择性蛋白精氨酸甲基转移酶 4 (PRMT4; CARM1) 抑制剂 (IC50<10 nM)。
| Cas No. | 2080306-20-1 |
| 化学名 | N-methyl-N-[[2-[1-[2-(methylamino)ethyl]-4-piperidinyl]-4-pyridinyl]methyl]-3-phenoxy-benzamide |
| Canonical SMILES | O=C(N(CC1=CC(C2CCN(CCNC)CC2)=NC=C1)C)C3=CC=CC(OC4=CC=CC=C4)=C3 |
| 分子式 | C28H34N4O2 |
| 分子量 | 458.6 |
| 溶解度 | 30mg/mL in ethanol, or in DMSO, or in DMF |
| 储存条件 | Store at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
| 产品描述 | TP-064 is a potent inhibitor of protein arginine methyltransferase 4 (PRMT4; IC50 in vitro. For more information on TP-064 please visit the Structural Genomics Consortium (SGC). The negative control, TP-064N, for TP-064 is also available exclusively through the SGC. You can submit a request to receive the negative control here. |
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