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A2aR/A2bR antagonist-1
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
A2aR/A2bR antagonist-1图片
CAS NO:2239273-34-6
包装与价格:
包装价格(元)
10mM (in 1mL DMSO)电议
5mg电议
10mg电议
25mg电议
50mg电议
100mg电议
200mg电议
500mg电议

产品介绍
A2aR/A2bR 拮抗剂-1 是一种口服生物可利用的选择性双重腺苷受体 (A2aR/A2bR) 拮抗剂。
Cas No.2239273-34-6
Canonical SMILESN#CC1=CC=CC(C2=NC(N)=NC(C3=CN(CC4=NC(C(C)(O)C)=CC=C4)N=N3)=C2)=C1C
分子式C23H22N8O
分子量426.47
溶解度DMSO: 250 mg/mL (586.21 mM)
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

A2aR/A2bR antagonist-1 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist with immunomodulatory activity[1].

[1]. Seitz L, et al. Safety, tolerability, and pharmacology of AB928, a novel dual adenosine receptor antagonist, in a randomized, phase 1 study in healthy volunteers. Invest New Drugs. 2019 Aug;37(4):711-721.