TAK-960
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
包装与价格:
包装 | 价格(元) |
5mg | 电议 |
10mg | 电议 |
50mg | 电议 |
100mg | 电议 |
产品介绍
CAS: | 1137868-52-0 |
分子式: | C27H34F3N7O3 |
分子量: | 561.60 |
纯度: | >98% |
溶解性: | DMSO |
存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
研究领域: | Cancer |
Target: | 0.8 nM (IC50)-PLK1,16.9 nM (IC50)-PLK2,50.2 nM (IC50)-PLK3,19.6 nM (IC50)-FAK/PTK2,25.6 nM (IC50)-MLCK/MYLK,58.2 nM (IC50)-FES/FPS |
描述: | TAK-960 is an orally available, selective inhibitor of polo-like kinase 1 (PLK1), with an IC50 of 0.8 nM at 10 μM ATP; TAK-960 also shows inhibitory activities against PLK2 and PLK3, with IC50s of 16. |