产品名称: | 马来酸罗格列酮 |
CAS: | 155141-29-0 |
分子式: | C22H23N3O7S |
分子量: | 473.50 |
纯度: | ≥98% |
溶解性: | DMSO |
存储: | Powder -20℃ 3 years; 4℃ 2 years In solvent -80℃ 6 months;-20℃ 1 month |
研究领域: | Metabolic Disease/Inflammation/Immunology |
Target: | EC50: 30 nM (PPARγ1), 100 nM (PPARγ2)[1], 60 nM (PPARγ)[2], appr 30 nM (TRPC5)[4]Kd: appr 40 nM (PPARγ)[1]IC50: appr 22.5 μM (TRPM2)[4] |
描述: | Rosiglitazone maleate is a potent and selective activator of PPARγ, with EC50 of 30 nM, 100 nM and 60 nM for PPARγ1, PPARγ2, and PPARγ, respectively, and a Kd of appr 40 nM for PPARγ; Rosiglitazone ma |