CAS NO: | 2416022-90-5 |
包装 | 价格(元) |
5mg | 电议 |
10mg | 电议 |
50mg | 电议 |
100mg | 电议 |
生物活性 | DDR1-IN-5 is a selectiveDiscoidin Domain Receptorfamily, member 1 (DDR1)inhibitor with anIC50of 7.36 nM. DDR1-IN-5 inhibits auto-phosphorylation DDR1b (Y513) with anIC50of 4.1 nM. DDR1-IN-5 has anti-cancer activity[1]. | ||||||||||||||||
IC50& Target[1] |
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体外研究 (In Vitro) | DDR1-IN-5 (compound 121; for 24 hours) inhibits collagen production in human hepatic stellate cell LX-2 (IC50=62 nM)[1]. | ||||||||||||||||
分子量 | 434.37 | ||||||||||||||||
性状 | Solid | ||||||||||||||||
Formula | C22H13F3N6O | ||||||||||||||||
CAS 号 | 2416022-90-5 | ||||||||||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||||||||||
储存方式 | 4°C, sealed storage, away from moisture and light *In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light) | ||||||||||||||||
溶解性数据 | In Vitro: DMSO : 2.78 mg/mL(6.40 mM;ultrasonic and warming and heat to 60℃) 配制储备液
* 请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 |