CAS NO: | 1314796-00-3 |
包装 | 价格(元) |
10 mM * 1 mL in DMSO | 电议 |
5mg | 电议 |
10mg | 电议 |
25mg | 电议 |
50mg | 电议 |
100mg | 电议 |
200mg | 电议 |
生物活性 | HGPR91 antagonist 1 is a potent and selective small moleculehGPR91antagonist with anIC50of 7 μM[1]. | ||||||||||||||||
IC50& Target | IC50: 7 μM (HGPR91)[1] | ||||||||||||||||
体内研究 (In Vivo) | HGPR91 antagonist 1 leads to 59, 76% inhibition of ΔMAP at 2, 4 hours and has shown rat plasma protein binding 99%. HGPR91 antagonist 1 has engaged the target under the in vivo condition. HGPR91 antagonist 1 has clearance (CL) of 0.2 nmol/min/mg of RLM[1].
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分子量 | 529.53 | ||||||||||||||||
性状 | Solid | ||||||||||||||||
Formula | C31H23F4N3O | ||||||||||||||||
CAS 号 | 1314796-00-3 | ||||||||||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||||||||||
储存方式 |
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溶解性数据 | In Vitro: DMSO : ≥ 125 mg/mL(236.06 mM) *"≥" means soluble, but saturation unknown. 配制储备液
* 请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 |