L-R4W2 是香草素受体 1 (VR1, TRPV1) 的有效拮抗剂，IC50 为 0.1 μM。
| Cas No. | 206350-79-0 |
| 化学名 | (S,Z)-2-amino-N-((6S,7Z,9S,10Z,12S,13Z,15S,16Z,18S)-15,18-bis((1H-indol-3-yl)methyl)-1-amino-9,12-bis(3-guanidinopropyl)-7,10,13,16,19-pentahydroxy-1,19-diimino-2,8,11,14,17-pentaazanonadeca-7,10,13,16-tetraen-6-yl)-5-guanidinopentanimidic acid |
| Canonical SMILES | N[C@@](/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/[C@@](C(O)=N)([H])CC1=CNC2=CC=CC=C12)([H])CC3=CNC4=CC=CC=C34)([H])CCCNC(N)=N)([H])CCCNC(N)=N)([H])CCCNC(N)=N)([H])CCCNC(N)=N |
| 分子式 | C46H71N21O6 |
| 分子量 | 1014.2 |
| 溶解度 | Soluble to 1 mg/ml in Water |
| 储存条件 | Desiccate at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
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