CYP1B1-IN-5 (Compound 6q) 是一种有效的、选择性的细胞色素 P450 1B1 (CYP1B1) 抑制剂，IC50为 4.7 nM。
| 生物活性 | CYP1B1-IN-5 (Compound 6q) is a potent and selectivecytochrome P4501B1 (CYP1B1) inhibitor with anIC50of 4.7 nM[1]. |
| IC50& Target[1] | CYP1B1 4.7 nM (IC50) | CYP1A1 190.7 nM (IC50) | CYP1A2 585.7 nM (IC50) |
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体外研究
(In Vitro) | CYP1B1-IN-5 (Compound 6q) 通过与残基 Phe231、Phe134 和血红素形成 π-π 叠加相互作用，与 CYP1B1 的结合口袋结合[1]。
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
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