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XZ426
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
XZ426图片
CAS NO:1638504-52-5
包装与价格:
包装价格(元)
5mg电议
10mg电议
25mg电议
50mg电议
100mg电议

产品介绍
XZ426 是一种有效的整合酶链转移抑制剂,具有抗HIV活性。
生物活性

XZ426 is a potent integrase strand transfer inhibitor with anti-HIVactivity[1].

体外研究
(In Vitro)

Intasomes are the target of the latest generation of antiretroviral drugs, integrase (IN) strand transfer inhibitors (INSTI). To better understand how INSTIs interact with HIV intasomes, we assembled the complex with bictegravir (BIC), the leading second-generation INSTI and the most broadly effective of all clinically approved INSTIs. Among these, XZ426 is a lead candidate that has shown superior efficacy to all clinically used and developed compounds against known drug-resistant variants[1].

分子量

446.45

性状

Solid

Formula

C22H24F2N4O4

CAS 号

1638504-52-5

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式
Powder-20°C3 years
4°C2 years
In solvent-80°C6 months
-20°C1 month