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Theodrenaline((±)-Theodrenaline)
本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。
Theodrenaline((±)-Theodrenaline)图片
CAS NO:13460-98-5
包装与价格：
包装价格(元)
1mg电议
5mg电议
10mg电议
20mg电议

产品介绍
Theodrenaline ((±)-Theodrenaline) 是一种心脏兴奋剂，也可与咖啡碱一起用作抗低血压剂。
Cas No.13460-98-5
别名茶碱那林; (±)?-?Theodrenaline
Canonical SMILESO=C(N1C)N(C)C2=C(N(CCNCC(C3=CC=C(O)C(O)=C3)O)C=N2)C1=O
分子式C17H21N5O5
分子量375.38
溶解度Soluble in DMSO
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

Theodrenaline is a cardiac stimulant, also acts as an anti-hypotensive agent together with cafedrine.

Akrinor evokes a positive inotropic effect in human atrial trabeculae via stimulation of β-adrenoceptors (AR)[1].

AkrinorTM produces significant potentiation of FSK effects, conceivable by PDE-inhibition, only at very high, clinically irrelevant concentrations of 420 mg/L[1].

[1]. Kloth B, et al. AkrinorTM, a Cafedrine/ Theodrenaline Mixture (20:1), Increases Force of Contraction of Human Atrial Myocardium But Does Not Constrict Internal Mammary Artery In Vitro. Front Pharmacol. 2017 May 23;8:272.