GSK1940029

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GSK1940029

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

1150701-66-8

包装与价格：

包装	价格(元)
10 mM * 1 mL in DMSO	电议
5mg	电议
10mg	电议
50mg	电议
100mg	电议
200mg	电议

产品名称

SCD inhibitor 1

产品介绍

GSK1940029 (SCD inhibitor 1) 是一种有效的酰基-辅酶A去饱和酶 (SCD) 抑制剂，详细信息请参考专利 WO/2009060053 A1 中的化合物 example 16。

生物活性

GSK1940029 (SCD inhibitor 1) is astearoyl-coa desaturase(SCD) inhibitor extracted from patent WO/2009060053 A1, compound example 16.

IC₅₀& Target

Stearoyl-CoA Desaturase (SCD)^[1]

体外研究
(In Vitro)

GSK1940029 (SCD inhibitor 1) is a stearoyl-coa desaturase (SCD), which can be used to treat and/or preventing various diseases, including those mediated by SCD enzyme, such as diseases related to elevated lipid levels, cardiovascular disease, diabetes, obesity, metabolic syndrome, skin disorders such as acne, diseases or conditions related to cancer and the treatment of symptoms linked to the production of the amyloid plaque-forming Aβ42 peptide such as Alzheimer's disease^[1].

Clinical Trial

分子量

391.25

性状

Solid

Formula

C₁₈H₁₆Cl₂N₄O₂

CAS 号

1150701-66-8

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Powder	-20°C	3 years
	4°C	2 years
In solvent	-80°C	6 months
	-20°C	1 month

溶解性数据

In Vitro:

DMSO : ≥ 32 mg/mL(81.79 mM)

*"≥" means soluble, but saturation unknown.

配制储备液

浓度溶剂体积质量

1 mg

5 mg

10 mg

1 mM	2.5559 mL	12.7796 mL	25.5591 mL
5 mM	0.5112 mL	2.5559 mL	5.1118 mL
10 mM	0.2556 mL	1.2780 mL	2.5559 mL

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80℃, 6 months; -20℃, 1 month。-80℃ 储存时，请在 6 个月内使用，-20℃ 储存时，请在 1 个月内使用。