CAS NO: | 357399-43-0 |
包装 | 价格(元) |
5mg | 电议 |
10mg | 电议 |
50mg | 电议 |
生物活性 | Bupropion morpholinol (Hydroxy Bupropion) is a major metabolite of Bupropion. Bupropion morpholinol inhibitsDopamine,Norepinephrine transportersand theα4β2 nicotinic receptorin vitro. Bupropion morpholinol contributes to antidepressant and smoking cessation activities[1][2][3]. | ||||||||||||||||
IC50& Target | Dopamine transporter[2], Norepinephrine transporter[2], α4β2 nicotinic receptor[2] | ||||||||||||||||
体外研究 (In Vitro) | Bupropion morpholinol is produced from Bupropion by the genetically polymorphic enzyme CYP2B6 in vivo[1]. | ||||||||||||||||
分子量 | 255.74 | ||||||||||||||||
性状 | Solid | ||||||||||||||||
Formula | C13H18ClNO2 | ||||||||||||||||
CAS 号 | 357399-43-0 | ||||||||||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||||||||||
储存方式 | -20°C, sealed storage, away from moisture *In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture) | ||||||||||||||||
溶解性数据 | In Vitro: DMSO : 20 mg/mL(78.20 mM;Need ultrasonic and warming) Ethanol : 20 mg/mL(78.20 mM;Need ultrasonic and warming) 配制储备液
* 请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 |