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Cyclosporin A-d4
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Cyclosporin A-d4图片
包装与价格:
包装价格(元)
1mg电议
5mg电议

产品名称
Cyclosporine A-d4
Ciclosporin A-d4
CsA-d4
产品介绍
Cyclosporin A-d4 是 Cyclosporin A 的氘代物。 Cyclosporin A (Cyclosporine A) 是一种免疫抑制剂,能与亲环素结合,抑制calcineurin活性的IC50值为 7 nM。Cyclosporin A 也抑制CD11a/CD18粘附分子。
生物活性

Cyclosporin A-d4 is the deuterium labeled Cyclosporin A. Cyclosporin A (Cyclosporine A) is an immunosuppressant which binds to the cyclophilin and inhibitsphosphataseactivity of calcineurin with an IC50 of 5 nM. Cyclosporin A also inhibits CD11a/CD18 ad

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

分子量

1206.64

Formula

C62H107D4N11O12

中文名称

环孢霉素A d4;环孢素A d4;环孢多肽A d4;环孢灵 d4;赛斯平 d4;环孢素 d4

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.