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Artemotil(&beta-Arteether)
本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。
Artemotil(&beta-Arteether)图片
CAS NO:75887-54-6
包装与价格：
包装价格(元)
10mM (in 1mL DMSO)电议
5mg电议
10mg电议
50mg电议
100mg电议

产品介绍
Artemotil (β-Arteether) (β-Arteether) 具有抗疟活性，用于治疗耐氯喹的恶性疟原虫疟疾，IC50 为 1.61 nM。
Cas No.75887-54-6
别名蒿乙醚; β-Arteether; (+)-Arteether; Arteether
Canonical SMILESC[C@@H]1[C@@](CC[C@@H](C)[C@]2([H])CC[C@]3(C)O4)([H])[C@@]2(OO3)[C@]4([H])O[C@@H]1OCC
分子式C17H28O5
分子量312.4
溶解度DMSO : 50 mg/mL (160.05 mM);Water :< 0.1 mg/mL (insoluble)
储存条件Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

Artemotil (β-Arteether) is a fast acting blood schizonticide specifically indicated for the treatment of chloroquine-resistant Plasmodium falciparum malaria and cerebral malaria cases. Target:Artemotil is a semi-synthetic derivative of artemisinin, a natural product of the Chinese plant Artemisia annua.

[1]. Looareesuwan S, et al. Dose-finding and efficacy study for i.m. artemotil (beta-arteether) and comparison with i.m. artemether in acute uncomplicated P. falciparum malaria. Br J Clin Pharmacol. 2002 May;53(5):492-500.