Macbecin 是一种稳定的HSP90抑制剂,与 ATP 结合位点结合,IC50为 2 μM,Kd为 0.24 μM。Macbecin 具有抗肿瘤活性和细胞毒性。
生物活性 | Macbecin is a stableHSP90inhibitor by binding to the ATP-binding site with anIC50of 2 μM and aKdof 0.24 μM. Macbecin exhibits antitumor and cytocidal activities[1]. |
IC50& Target | HSP90 2 μM (IC50) | HSP90 0.24 μM (Kd) |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |