(R)-HH2853 是一种突变型EZH2抑制剂,对EZH2-Y641F的IC50<100 nM。(R)-HH2853 可用于癌症和自身免疫性疾病 (WO2018045971A1; compound 201)。
生物活性 | (R)-HH2853 is amutantEZH2inhibitor with anIC50of<100 nm forEZH2-Y641F. (R)-HH2853 can be used forcancerand autoimmune diseases (WO2018045971A1; compound 201)[1]. |
IC50& Target[1] | EZH2 Y641F mutant type <100 nM (IC50) |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |