MJ 15 是一种有效的选择性 CB1 受体拮抗剂,对大鼠 CB1 受体的 Ki 为 27.2 pM,IC50 为 118.9 pM。
Cas No. | 944154-76-1 |
化学名 | (Z)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carbimidic acid |
Canonical SMILES | CC(C(/C(O)=N/CC1=CN=CC=C1)=NN2C3=C(Cl)C=C(Cl)C=C3)=C2C4=CC=C(Cl)C=C4 |
分子式 | C23H17Cl3N4O |
分子量 | 471.77 |
溶解度 | DMSO:<100 mM,Ethanol: slightly soluble |
储存条件 | Store at RT |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |