CAS NO: | 1782228-83-4 |
包装 | 价格(元) |
100mg | 电议 |
250mg | 电议 |
500mg | 电议 |
生物活性 | ST1936 oxalate is a selective, nanomolar affinity5-HT6receptoragonist withKivalues of 13 nM, 168 nM and 245 nM for human5-HT6, 5-HT7and 5-HT2Breceptors, respectively. ST1936 oxalate also shows moderate affinity (Kiof 300 nM) for human and ratα2adrenergic receptor[1]. | ||||||
IC50& Target[1] |
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体外研究 (In Vitro) | ST1936 oxalate appears to be relatively selective for 5-HT6receptors, although it has shown affinity also for 5-HT2B, 5-HT1A, 5-HT7receptor and α-adrenergic receptors when tested in a broad crossreactivity panel that comprised G-protein-coupled receptors, ion channel binding sites, enzymes, and transporters[1]. | ||||||
体内研究 (In Vivo) | ST1936 (5, 10, 20 mg/kg; i.p.) oxalate increases in a dose dependent manner extracellular dopamine (DA) and NA levels in the prefrontal cortex (PFCX)[2]. | ||||||
分子量 | 326.78 | ||||||
Formula | C15H19ClN2O4 | ||||||
CAS 号 | 1782228-83-4 | ||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |