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Nexopamil racemate
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Nexopamil racemate图片
CAS NO:116759-35-4
包装与价格:
包装价格(元)
100mg电议
250mg电议
500mg电议

产品名称
奈索帕米
产品介绍
Nexopamil racemate 是 Nexopamil 的外消旋体。Nexopamil 是体内血栓形成和体外血小板聚集中的一种联合Ca2+/5-HT2拮抗剂。
生物活性

Nexopamil racemate is the racemate of Nexopamil. Nexopamil is a combinedCa2+/5-HT2antagonist on thrombus formation in vivo and on platelet aggregation in vitro.

IC50& Target

5-HT2Receptor

 

体外研究
(In Vitro)

Serotonin-induced platelet aggregation in dog platelet-rich plasma (PRP) in vitro is most potently inhibited by Nexopamil (IC5081 nM)[1].

体内研究
(In Vivo)

Nexopamil (0.05 mg/kg) completely abolishes cyclic flow reductions (CFRs) during the first 30 min after application without significantly altering hemodynamics[1].

分子量

404.59

Formula

C24H40N2O3

CAS 号

116759-35-4

中文名称

奈索帕米

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.