| CAS NO: | 1092502-33-4 |
| 包装 | 价格(元) |
| 100mg | 电议 |
| 250mg | 电议 |
| 500mg | 电议 |
| 生物活性 | GW 833972A is a selectiveCB2receptoragonist. GW 833972A inhibits induced nerve depolarization and citric acid-induced cough in animal models[1]. | ||
| IC50& Target[1] |
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| 体外研究 (In Vitro) | GW 833972A (0.3-300 μM; 10 min) 抑制辣椒素诱导的人和豚鼠去极化，还抑制前列腺素 E(2) 和高渗盐水诱导的豚鼠离体迷走神经去极化[1]。 | ||
| 体内研究 (In Vivo) | GW 833972A (30 mg/kg, 2 mL/kg;腹腔注射; 单次剂量, 试验开始前 30 min 注射) 能够抑制柠檬酸诱导的有意识豚鼠的咳嗽症状。它还抑制辣椒素引起的主支气管血浆蛋白渗出现象[1]。 | ||
| 分子量 | 444.24 | ||
| Formula | C18H14Cl2F3N5O | ||
| CAS 号 | 1092502-33-4 | ||
| 运输条件 | Room temperature in continental US; may vary elsewhere. | ||
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
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