L-365,260 是一种具有口服活性的选择性非肽胃泌素和脑胆囊收缩素受体 (CCK-B) 拮抗剂,Kis 分别为 1.9 nM 和 2.0 nM。
Cas No. | 118101-09-0 |
化学名 | (R)-1-(1-methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-(m-tolyl)urea |
Canonical SMILES | O=C1N(C)C2=CC=CC=C2C(C3=CC=CC=C3)=N[C@H]1NC(NC4=CC=CC(C)=C4)=O |
分子式 | C24H22N4O2 |
分子量 | 398.46 |
溶解度 | <39.85mg/ml in DMSO;<39.85mg/ml in ethanol |
储存条件 | Store at -20℃ |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |