JTP-117968 是选择性的糖皮质激素受体调节剂 (非甾类的 SGRM，IC50值为 6.8 nM)，具有改善的转录抑制/转激活解离活性。
| 生物活性 | JTP-117968, a novel selectiveglucocorticoid receptormodulator (a non-steroidal SGRM,IC50of 6.8 nM), exhibits improved transrepression/transactivation dissociation[1]. |
体外研究
(In Vitro) | JTP-117968 has partial TR activity, but exhibits extremely low TA activity[1].
|
| 分子量 | |
| Formula | |
| CAS 号 | |
| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
m.cnreagent.com
