L-168,049 是一种有效的、选择性的、具有口服活性的非竞争性胰高血糖素受体拮抗剂,对人、鼠和犬胰高血糖素受体的 IC50 分别为 3.7 nM、63 nM 和 60 nM。
Cas No. | 191034-25-0 |
化学名 | 4-(3-(5-bromo-2-propoxyphenyl)-5-(4-chlorophenyl)-1H-pyrrol-2-yl)pyridine |
Canonical SMILES | BrC1=CC=C(C(C2=C(C3=CC=NC=C3)NC(C(C=C4)=CC=C4Cl)=C2)=C1)OCCC |
分子式 | C24H20BrClN2O |
分子量 | 467.79 |
溶解度 | <46.78mg/ml in DMSO;<46.78mg/ml in ethanol |
储存条件 | Store at RT |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |